Cerebrolysin (Cerebrolysin®)

Neuropeptide Preparation | Neurological Recovery

Weight: Variable
Half-life: Minutes (component-dependent; e.g., BDNF ~10 min)
Chain: Multiple peptides
5 studies
2023 latest
3 recent
Well Studied
Dose 10-50mL depending on indication (stroke/TBI higher doses)
Frequency Once daily for acute conditions; 5 days weekly for chronic conditions
Cycle 7-30 days depending on condition (stroke/TBI 10-30 days, dementia 4 weeks)
Storage Room temperature ≤25°C, protected from light in original carton - never freeze

Community Research

Join others researching Cerebrolysin — share findings, ask questions, and learn from real experiences

Standardized neuropeptide preparation containing bioactive peptides and amino acids exhibiting neurotrophic and neuroprotective properties for stroke recovery, traumatic brain injury, and cognitive enhancement. Used clinically in 50+ countries.

Mechanism of Action

IV/IM administration provides optimal bioavailability and brain penetration of neuropeptides and neurotrophic factors.

01 Direct brain delivery
02 Standardized dosing
03 Extensive clinical evidence
04 Ready-to-use formulation
05 Used clinically in 50+ countries

Molecular Data

Molecular Weight
Variable
Chain Length
Multiple peptides
Type
Purified porcine brain proteins
Amino Acid Sequence
Bioactive peptide mixture

Complex or non-standard sequence format

Peak 0.0 mcg
Trough 0.0 mcg
SS Peak 0.0 mcg
SS Trough 0.0 mcg

Research Indications

Cognitive
Alzheimer's Disease moderate

Meta-analyses show modest cognitive improvements, though clinical significance remains debated.

Vascular Dementia effective

Multiple RCTs demonstrate significant ADAS-cog and CIBIC+ improvements.

Post-Stroke Cognitive Recovery moderate

Large meta-analysis shows significant NIHSS improvements; other studies found no functional benefit.

Neuroprotection
Acute Stroke moderate

Largest meta-analysis (1,879 patients) shows NIHSS benefits; independent analysis found no mRS improvement.

Traumatic Brain Injury most effective

Multiple trials including CAPTAIN series confirm GCS/GOS improvements.

Subarachnoid Hemorrhage moderate

Pilot trial shows promising 6-month outcomes; requires larger confirmatory studies.

Recovery
Motor Function Recovery moderate

Some studies show enhanced recovery; results vary significantly between trials.

Neurological Function effective

Early administration within 72 hours shows better outcomes than delayed treatment.

Dosing Protocols

Primary administration route with well-established protocols for direct brain delivery via IV/IM.

GoalDoseFrequencyRoute
Small Volume IVUp to 10mLOnce dailyUndiluted IV slow push over 3 minutes
IntramuscularUp to 5mLOnce dailyUndiluted IM injection over 3 minutes
Acute Stroke20-50mLOnce daily for 10-21 daysIV infusion (diluted to 100mL minimum)
Traumatic Brain Injury20-50mLOnce daily for 7-30 daysIV infusion (diluted to 100mL minimum)
Alzheimer's Disease10-30mL5 days weekly for 4 weeksIV injection/infusion (2-4 cycles yearly)
Vascular Dementia10-30mL5 days weekly for 4 weeksIV injection/infusion (2-4 cycles yearly)

Reconstitution Instructions

Materials Needed:
  • Cerebrolysin ampoules (5, 10, or 20 mL)
  • Saline, Ringer solution, or 5% glucose (minimum 100 mL for infusion)
  • Disposable one-way IV infusion sets and cannulas
  • Sterile syringes and alcohol swabs
  1. 1 Break ampoule and extract Cerebrolysin immediately before use
  2. 2 For direct injection: Up to 10 mL IV undiluted (slow 3 minutes) or 5 mL IM
  3. 3 For infusion: Dilute 10-50 mL to minimum 100 mL with compatible solution
  4. 4 Start infusion immediately after dilution—infuse within 15 minutes
  5. 5 Flush IV catheter with sodium chloride before and after administration
  6. 6 Use disposable one-way infusion sets; discard after use

Interactions

+
Piracetam
Safe combination with no significant interactions; both support cognitive function.
compatible
+
Donepezil
No interactions reported; may have synergistic cognitive effects in Alzheimer's treatment.
compatible
~
SSRIs
Potential additive neurotropic effects; monitor for enhanced antidepressant effects.
monitor
~
Tricyclic Antidepressants
May have additive neurological effects; requires careful monitoring.
monitor
!
Amino Acid Solutions
Contraindicated per prescribing information; do not mix in same infusion.
avoid
!
Cardiovascular Medications
Should not be mixed in same IV infusion per official guidelines.
avoid
!
Vitamin Solutions
Compatibility issues; do not mix in same IV infusion.
avoid
~
Noopept
Both enhance neurotrophic factors; potential additive effects—start with lower doses.
monitor

What to Expect

Week 1-2
Initial neuroprotective effects; possible mild side effects (dizziness, agitation)
Week 2-4
Neurological improvements become apparent; cognitive function may begin to improve
Week 4-8
Continued recovery; motor function improvements in stroke/TBI patients
Week 8-12
Sustained benefits; cognitive enhancement plateaus in chronic conditions

Side Effects & Safety

Common Side Effects

  • Generally well tolerated
  • Possible mild dizziness or agitation in early treatment

Stop Signs - Discontinue if:

  • Severe allergic reactions (anaphylaxis, severe rash)
  • New onset seizure activity
  • Significant cardiovascular events during administration
  • Severe renal dysfunction or worsening kidney function

Contraindications

  • Epilepsy
  • Severe renal insufficiency
  • History of severe allergic reactions to porcine products

Quality Checklist

Good Signs

  • Clear amber solution from reputable source
  • Room temperature storage ≤25°C
  • Protected from light in original carton
  • Authorized EVER Pharma distributor

Warning Signs

  • Some published studies have been retracted due to research misconduct; rely on independent meta-analyses

Bad Signs

  • Frozen product or improper storage—never freeze
  • Mixing with incompatible solutions (amino acids, vitamins, cardiovascular medications)

References

  • Efficacy and Safety of Cerebrolysin in Neurorecovery After Moderate-Severe Traumatic Brain Injury: Results from the CAPTAIN II Trial
    Muresanu DF, Florian S, et al.
    Neurological Sciences (2020)

    Phase IIIb/IV RCT: patients with GCS 7-12 received 50 mL Cerebrolysin daily for 10 days + two additional 10 mL cycles; confirmed beneficial effects on overall outcome after moderate-severe TBI.

  • Safety and Efficacy of Cerebrolysin in Early Post-Stroke Recovery: A Meta-Analysis of Nine Randomized Clinical Trials
    Bornstein NM, Guekht A, Vester J, et al.
    Neurological Sciences (2018)

    Meta-analysis of 1,879 stroke patients showed NIHSS superiority of Cerebrolysin (MW 0.60, P < 0.0001); NNT = 7.7 for clinically relevant early neurological improvement.

  • Cerebrolysin for Functional Recovery in Patients with Acute Ischemic Stroke: A Meta-Analysis of Randomized Controlled Trials
    Xue LX, Zhang T, Zhao YW, et al.
    International Journal of Neuroscience (2017)

    Meta-analysis of 1,779 patients found no significant benefit on mRS response (RR 1.33, P=0.28) or Barthel Index; concluded routine use for long-term stroke rehabilitation not supported.

  • Cerebrolysin in Patients with TBI: Systematic Review and Meta-Analysis
    Jarosz K, Kojder K, Andrzejewska A, Solek-Pastuszka J, Jurczak A
    Brain Sciences (2023)

    10 studies of 8,749 TBI patients; GOS improvement was statistically significant (mean difference 0.422, P = 0.000); mortality and length of stay were not significantly affected.

  • Cerebrolysin in Mild-to-Moderate Alzheimer's Disease: A Meta-Analysis of Randomized Controlled Clinical Trials
    Gauthier S, Proano JV, Jia J, et al.
    Dementia and Geriatric Cognitive Disorders (2015)

    6 RCTs in mild-to-moderate AD; Cerebrolysin significantly superior to placebo on ADAS-cog at 4 weeks (SMD -0.40, P=0.003) and CIBIC global clinical change at 4 weeks and 6 months.

Disclaimer

This information is for educational and research purposes only. Consult a healthcare professional before use.